Explore Targets
Showing 465 matching result(s) | Selected target(s): 0
| SELECT | TARGET ID | TARGET NAME | UNIPROT AC | UNIPROT ID | PANTHER CLASS | MAX PHASE | STRUCTURE INFO | SOURCE | STRUCTURE |
|---|---|---|---|---|---|---|---|---|---|
| D0001 | Arachidonate 5-lipoxygenase | P09917 | LOX5_HUMAN | oxygenase | Successful | Downloaded from PDB (6N2W) | 6N2W | ||
| D0002 | Diacylglycerol acyltransferase 1 | O75907 | DGAT1_HUMAN | acyltransferase | Successful | Downloaded from PDB (6VP0) | 6VP0 | ||
| D0003 | Caspase-1 | P29466 | CASP1_HUMAN | Undefined | Clinical trial | Downloaded from PDB (6F6R) | 6F6R | ||
| D0004 | PAK-4 protein kinase | O96013 | PAK4_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (5ZJW) | 5ZJW | ||
| D0005 | Thymidylate synthase | P04818 | TYSY_HUMAN | methyltransferase | Clinical trial | Downloaded from PDB (1HVY) | 1HVY | ||
| D0006 | Aggrecanase | Q9UNA0 | ATS5_HUMAN | metalloprotease | Clinical trial | Downloaded from PDB (3HYG) | 3HYG | ||
| D0007 | Presenilin 2 | P49810 | PSN2_HUMAN | aspartic protease | Clinical trial | Downloaded from PDB (7Y5X) | 7Y5X | ||
| D0008 | MAP kinase signal-integrating kinase 2 | Q9HBH9 | MKNK2_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (6CJ5) | 6CJ5 | ||
| D0009 | Metabotropic glutamate receptor 5 | P41594 | GRM5_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (6FFI) | 6FFI | ||
| D0010 | Gamma-secretase | Q96BI3+Q9NZ42+P49768+Q92542 | APH1A_HUMAN+APH1B_HUMAN+PEN2_HUMAN+NICA_HUMAN+PSN1_HUMAN | protease | Successful | Downloaded from PDB (7D8X) | 7D8X | ||
| D0011 | Carbonic anhydrase XII | O43570 | CAH12_HUMAN | dehydratase | Successful | Downloaded from PDB (6G5L) | 6G5L | ||
| D0012 | Dihydrofolate reductase | P00374 | DYR_HUMAN | reductase | Successful | Downloaded from PDB (1KMV) | 1KMV | ||
| D0013 | Matrix metalloproteinase-8 | P22894 | MMP8_HUMAN | metalloprotease | Clinical trial | Downloaded from PDB (4QKZ) | 4QKZ | ||
| D0014 | Voltage-gated potassium channel Kv1.5 | P22460 | KCNA5_HUMAN | voltage-gated ion channel | Successful | Modelled with AlphaFold (AF-P22460-F1-model_v4) | AB INITIO | ||
| D0015 | Urokinase-type plasminogen activator | P00749 | UROK_HUMAN | serine protease | Successful | Downloaded from PDB (1C5Y) | 1C5Y | ||
| D0016 | MEK kinase kinase 1 | Q92918 | M4K1_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (7R9N) | 7R9N | ||
| D0017 | Fyn tyrosine protein kinase | P06241 | FYN_HUMAN | non-receptor tyrosine protein kinase | Successful | Downloaded from PDB (2DQ7) | 2DQ7 | ||
| D0018 | Heat shock protein 90 alpha | P07900 | HS90A_HUMAN | Hsp90 family chaperone | Successful | Downloaded from PDB (5J2X) | 5J2X | ||
| D0019 | Melanin-concentrating hormone receptor 1 | Q99705 | MCHR1_HUMAN | G-protein coupled receptor | Clinical trial | Modelled with SWISS-MODEL (7E32.1.E) | HOMOLOGY | ||
| D0020 | S-mephenytoin 4-hydroxylase | P11712 | CP2C9_HUMAN | oxygenase | Successful | Downloaded from PDB (1R9O) | 1R9O | ||
| D0021 | Phosphodiesterase 4B | Q07343 | PDE4B_HUMAN | phosphodiesterase | Clinical trial | Downloaded from PDB (5OHJ) | 5OHJ | ||
| D0022 | Tumor necrosis factor | P01375 | TNFA_HUMAN | intercellular signal molecule | Successful | Downloaded from PDB (7JRA) | 7JRA | ||
| D0023 | Dopamine D3 receptor | P35462 | DRD3_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7CMV) | 7CMV | ||
| D0024 | Neuropeptide Y receptor type 2 | P49146 | NPY2R_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (7DDZ) | 7DDZ | ||
| D0025 | Voltage-gated potassium channel Kv11.1 | Q12809 | KCNH2_HUMAN | ion channel | Successful | Downloaded from PDB (5VA1) | 5VA1 | ||
| D0026 | Carbonic anhydrase II | P00918 | CAH2_HUMAN | dehydratase | Successful | Downloaded from PDB (3K34) | 3K34 | ||
| D0027 | Cyclin-dependent kinase 8 | P49336 | CDK8_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (5XS2) | 5XS2 | ||
| D0028 | Muscarinic acetylcholine receptor M4 | P08173 | ACM4_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (5DSG) | 5DSG | ||
| D0029 | Alpha-galactosidase A | P06280 | AGAL_HUMAN | galactosidase | Successful | Downloaded from PDB (6IBK) | 6IBK | ||
| D0030 | Norepinephrine transporter | P23975 | SC6A2_HUMAN | primary active transporter | Successful | Modelled with SWISS-MODEL (6VRH.1.A) | HOMOLOGY | ||
| D0031 | Cathepsin K | P43235 | CATK_HUMAN | cysteine protease | Clinical trial | Downloaded from PDB (4X6H) | 4X6H | ||
| D0032 | Toll-like receptor 9 | Q9NR96 | TLR9_HUMAN | transmembrane signal receptor | Clinical trial | Modelled with AlphaFold (AF-Q9NR96-F1-model_v4) | AB INITIO | ||
| D0033 | Dopamine D1 receptor | P21728 | DRD1_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7JVP) | 7JVP | ||
| D0034 | Glutamate receptor ionotropic NMDA 2A | Q12879 | NMDE1_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5H8Q) | 5H8Q | ||
| D0035 | Bacterial DNA gyrase | P20831+P0A0K8 | GYRA_STAAU+GYRB_STAAU | Undefined | Successful | Downloaded from PDB (6Z1A) | 6Z1A | ||
| D0036 | Progesterone receptor | P06401 | PRGR_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (1SQN) | 1SQN | ||
| D0037 | Janus kinase 3 | P52333 | JAK3_HUMAN | non-receptor tyrosine protein kinase | Successful | Downloaded from PDB (5LWM) | 5LWM | ||
| D0038 | Voltage-gated sodium channel alpha Nav1.7 | Q15858 | SCN9A_HUMAN | voltage-gated ion channel | Clinical trial | Downloaded from PDB (7W9K) | 7W9K | ||
| D0039 | G1/S-specific cyclin-D1 | P24385 | CCND1_HUMAN | kinase activator | Clinical trial | Downloaded from PDB (6P8E) | 6P8E | ||
| D0040 | Valosin-containing protein p97 | P55072 | TERA_HUMAN | primary active transporter | Clinical trial | Downloaded from PDB (7PUX) | 7PUX | ||
| D0041 | Endothelin A receptor | P25101 | EDNRA_HUMAN | Undefined | Successful | Downloaded from PDB (8HCQ) | 8HCQ | ||
| D0042 | Aryl hydrocarbon receptor | P35869 | AHR_HUMAN | basic helix-loop-helix transcription factor | Successful | Downloaded from PDB (7ZUB) | 7ZUB | ||
| D0043 | Protein-tyrosine phosphatase SHP-2 | Q06124 | PTN11_HUMAN | protein phosphatase | Clinical trial | Downloaded from PDB (7PPM) | 7PPM | ||
| D0044 | B2 bradykinin receptor | P30411 | BKRB2_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7F6I) | 7F6I | ||
| D0045 | Casein kinase I alpha | P48729 | KC1A_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (6GZD) | 6GZD | ||
| D0046 | AP endonuclease 1 | P27695 | APEX1_HUMAN | Undefined | Clinical trial | Downloaded from PDB (7TC2) | 7TC2 | ||
| D0047 | Endoplasmic reticulum to nucleus signaling 1 | O75460 | ERN1_HUMAN | tyrosine protein kinase receptor | Clinical trial | Downloaded from PDB (6W39) | 6W39 | ||
| D0048 | Oxysterols receptor LXR-beta | P55055 | NR1H2_HUMAN | C4 zinc finger nuclear receptor | Clinical trial | Downloaded from PDB (6S5K) | 6S5K | ||
| D0049 | Dopamine D4 receptor | P21917 | DRD4_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (5WIU) | 5WIU | ||
| D0050 | Tyrosine-protein kinase BTK | Q06187 | BTK_HUMAN | non-receptor tyrosine protein kinase | Successful | Downloaded from PDB (5P9J) | 5P9J | ||
| D0051 | Multidrug resistance protein 1 | P08183 | MDR1_HUMAN | ATP-binding cassette (ABC) transporter | Clinical trial | Downloaded from PDB (7A69) | 7A69 | ||
| D0052 | Sterol O-acyltransferase | P35610+O75908 | SOAT1_HUMAN+SOAT2_HUMAN | acyltransferase | Clinical trial | Downloaded from PDB (6L47) | 6L47 | ||
| D0053 | NAD-dependent deacetylase sirtuin-1 | Q96EB6 | SIR1_HUMAN | Undefined | Clinical trial | Downloaded from PDB (4I5I) | 4I5I | ||
| D0054 | Aldose reductase | P15121 | ALDR_HUMAN | reductase | Successful | Downloaded from PDB (4GCA) | 4GCA | ||
| D0055 | Induced myeloid leukemia cell differentiation protein Mcl-1 | Q07820 | MCL1_HUMAN | Undefined | Clinical trial | Downloaded from PDB (6UDV) | 6UDV | ||
| D0056 | Focal adhesion kinase 1 | Q05397 | FAK1_HUMAN | non-receptor tyrosine protein kinase | Clinical trial | Downloaded from PDB (6YOJ) | 6YOJ | ||
| D0057 | Cationic trypsinogen | P07477 | TRY1_HUMAN | serine protease | Successful | Downloaded from PDB (2RA3) | 2RA3 | ||
| D0058 | Cholesteryl ester transfer protein | P11597 | CETP_HUMAN | Undefined | Clinical trial | Downloaded from PDB (4EWS) | 4EWS | ||
| D0059 | Serotonin transporter | P31645 | SC6A4_HUMAN | primary active transporter | Successful | Downloaded from PDB (5I6X) | 5I6X | ||
| D0060 | Beta-site APP-cleaving enzyme 2 | Q9Y5Z0 | BACE2_HUMAN | protease | Clinical trial | Downloaded from PDB (7D5B) | 7D5B | ||
| D0061 | Tubulin beta-2 chain | Q13885 | TBB2A_HUMAN | tubulin | Successful | Modelled with SWISS-MODEL (6WVL.1.B) | HOMOLOGY | ||
| D0062 | GABA A receptor gamma-3 | Q99928 | GBRG3_HUMAN | ligand-gated ion channel | Successful | Modelled with SWISS-MODEL (6HUG.1.C) | HOMOLOGY | ||
| D0063 | Muscarinic acetylcholine receptor M1 | P11229 | ACM1_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6ZFZ) | 6ZFZ | ||
| D0064 | Signal transducer and activator of transcription 3 | P40763 | STAT3_HUMAN | Rel homology transcription factor | Successful | Downloaded from PDB (6NJS) | 6NJS | ||
| D0065 | Pyruvate dehydrogenase kinase 1 | Q15118 | PDK1_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (2Q8G) | 2Q8G | ||
| D0066 | Adrenergic receptor alpha-1B | P35368 | ADA1B_HUMAN | G-protein coupled receptor | Successful | Modelled with AlphaFold (AF-P35368-F1-model_v4) | AB INITIO | ||
| D0067 | Dipeptidyl peptidase 8 | Q6V1X1 | DPP8_HUMAN | serine protease | Clinical trial | Downloaded from PDB (7OR4) | 7OR4 | ||
| D0068 | Acetylcholinesterase | P22303 | ACES_HUMAN | esterase | Successful | Downloaded from PDB (4M0E) | 4M0E | ||
| D0069 | Sodium/glucose cotransporter 2 | P31639 | SC5A2_HUMAN | secondary carrier transporter | Successful | Downloaded from PDB (7VSI) | 7VSI | ||
| D0070 | C-C chemokine receptor type 1 | P32246 | CCR1_HUMAN | cell adhesion molecule | Clinical trial | Downloaded from PDB (7VL8) | 7VL8 | ||
| D0071 | Trypanosoma Cruzipain | P25779 | CYSP_TRYCR | Undefined | Successful | Downloaded from PDB (1ME3) | 1ME3 | ||
| D0072 | Nitric-oxide synthase brain | P29475 | NOS1_HUMAN | oxidoreductase | Clinical trial | Downloaded from PDB (5VV0) | 5VV0 | ||
| D0073 | Leukotriene A-4 hydrolase | P09960 | LKHA4_HUMAN | Undefined | Successful | Downloaded from PDB (3U9W) | 3U9W | ||
| D0074 | Histamine H2 receptor | P25021 | HRH2_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7UL3) | 7UL3 | ||
| D0075 | Rotamase Pin1 | Q13526 | PIN1_HUMAN | chaperone | Clinical trial | Downloaded from PDB (3I6C) | 3I6C | ||
| D0076 | 5-HT 2B receptor | P41595 | 5HT2B_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7SRQ) | 7SRQ | ||
| D0077 | Protein-tyrosine phosphatase 1B | P18031 | PTN1_HUMAN | protein phosphatase | Clinical trial | Downloaded from PDB (7MNA) | 7MNA | ||
| D0078 | Apoptosis regulator Bcl-2 | P10415 | BCL2_HUMAN | Undefined | Successful | Downloaded from PDB (6GL8) | 6GL8 | ||
| D0079 | Dipeptidyl peptidase 4 | P27487 | DPP4_HUMAN | serine protease | Successful | Downloaded from PDB (4A5S) | 4A5S | ||
| D0080 | Phospholipase A2 | P04054 | PA21B_HUMAN | phospholipase | Successful | Downloaded from PDB (3ELO) | 3ELO | ||
| D0081 | 5-HT 6 receptor | P50406 | 5HT6R_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (7YS6) | 7YS6 | ||
| D0082 | Lysine-specific histone demethylase 1 | O60341 | KDM1A_HUMAN | oxidase | Clinical trial | Downloaded from PDB (2Z3Y) | 2Z3Y | ||
| D0083 | X-linked inhibitor of apoptosis protein | P98170 | XIAP_HUMAN | protease inhibitor | Clinical trial | Downloaded from PDB (4KJU) | 4KJU | ||
| D0084 | Protein arginine methyltransferase 1 | Q99873 | ANM1_HUMAN | protein modifying enzyme | Clinical trial | Downloaded from PDB (6NT2) | 6NT2 | ||
| D0085 | Carbonic anhydrase XIV | Q9ULX7 | CAH14_HUMAN | dehydratase | Successful | Downloaded from PDB (5CJF) | 5CJF | ||
| D0086 | 5-HT 2A receptor | P28223 | 5HT2A_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7WC8) | 7WC8 | ||
| D0087 | DNA topoisomerase II alpha | P11388 | TOP2A_HUMAN | DNA metabolism protein | Clinical trial | Downloaded from PDB (5GWK) | 5GWK | ||
| D0088 | Menin-MLL1 interaction | O00255+Q03164 | MEN1_HUMAN-KMT2A_HUMAN | Undefined | Clinical trial | Downloaded from PDB (4GQ4) | 4GQ4 | ||
| D0089 | Steryl-sulfatase | P08842 | STS_HUMAN | hydrolase | Successful | Downloaded from PDB (8EG3) | 8EG3 | ||
| D0090 | Vitamin D3 receptor | P11473 | VDR_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (3B0T) | 3B0T | ||
| D0091 | Neuronal acetylcholine receptor alpha-7 | P36544 | ACHA7_HUMAN | ligand-gated ion channel | Successful | Downloaded from PDB (5AFN) | 5AFN | ||
| D0092 | Monoglyceride lipase | Q99685 | MGLL_HUMAN | phospholipase | Clinical trial | Downloaded from PDB (3PE6) | 3PE6 | ||
| D0093 | Prostaglandin E2 receptor EP4 | P35408 | PE2R4_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (5YWY) | 5YWY | ||
| D0094 | Group IIA phospholipase A2 | P14555 | PA2GA_HUMAN | phospholipase | Clinical trial | Downloaded from PDB (5G3N) | 5G3N | ||
| D0095 | Integrin alpha-L | P20701 | ITAL_HUMAN | integrin | Successful | Downloaded from PDB (2ICA) | 2ICA | ||
| D0096 | Melanocortin receptor 1 | Q01726 | MSHR_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7F4H) | 7F4H | ||
| D0097 | Proteinase activated receptor 1 | P25116 | PAR1_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (3VW7) | 3VW7 | ||
| D0098 | Cannabinoid receptor 2 | P34972 | CNR2_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6KPC) | 6KPC | ||
| D0099 | Phosphoinositide dependent protein kinase-1 | O15530 | PDPK1_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (5LVO) | 5LVO | ||
| D0100 | Hypoxia-inducible factor 2 alpha | Q99814 | EPAS1_HUMAN | basic helix-loop-helix transcription factor | Successful | Downloaded from PDB (4GHI) | 4GHI | ||
| D0101 | MAPK-activated protein kinase 2 | P49137 | MAPK2_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (3M2W) | 3M2W | ||
| D0102 | Voltage-gated calcium channel alpha Cav2.2 | Q00975 | CAC1B_HUMAN | voltage-gated ion channel | Successful | Downloaded from PDB (7VFU) | 7VFU | ||
| D0103 | Prostaglandin E2 receptor EP2 | P43116 | PE2R2_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7CX2) | 7CX2 | ||
| D0104 | Voltage-gated sodium channel alpha Nav1.5 | Q14524 | SCN5A_HUMAN | voltage-gated ion channel | Successful | Downloaded from PDB (6LQA) | 6LQA | ||
| D0105 | Glucocorticoid receptor | P04150 | GCR_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (4UDD) | 4UDD | ||
| D0106 | Proto-oncogene c-Met | P08581 | MET_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (3DKC) | 3DKC | ||
| D0107 | Histone deacetylase 6 | Q9UBN7 | HDAC6_HUMAN | Undefined | Clinical trial | Downloaded from PDB (5WPB) | 5WPB | ||
| D0108 | Gastrin/cholecystokinin type B receptor | P32239 | GASR_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7F8W) | 7F8W | ||
| D0109 | Xanthine dehydrogenase/oxidase | P47989 | XDH_HUMAN | oxidoreductase | Successful | Downloaded from PDB (2CKJ) | 2CKJ | ||
| D0110 | Adrenergic receptor alpha-2B | P18089 | ADA2B_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6K41) | 6K41 | ||
| D0111 | Glutamate receptor AMPA 2 | P42262 | GRIA2_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5ZG2) | 5ZG2 | ||
| D0112 | Coagulation factor VII | P08709 | FA7_HUMAN | serine protease | Successful | Downloaded from PDB (5PAG) | 5PAG | ||
| D0113 | Voltage-gated sodium channel alpha Nav1.8 | Q9Y5Y9 | SCNAA_HUMAN | voltage-gated ion channel | Successful | Downloaded from PDB (7WE4) | 7WE4 | ||
| D0114 | Adrenergic receptor beta-1 | P08588 | ADRB1_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7BVQ) | 7BVQ | ||
| D0115 | Tissue-type plasminogen activator | P00750 | TPA_HUMAN | serine protease | Successful | Downloaded from PDB (1BDA) | 1BDA | ||
| D0116 | Proto-oncogene c-RAF | P04049 | RAF1_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (3OMV) | 3OMV | ||
| D0117 | Muscarinic acetylcholine receptor M2 | P08172 | ACM2_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (3UON) | 3UON | ||
| D0118 | Opioid receptor sigma 1 | Q99720 | SGMR1_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5HK1) | 5HK1 | ||
| D0119 | Poly [ADP-ribose] polymerase 1 | P09874 | PARP1_HUMAN | DNA metabolism protein | Successful | Downloaded from PDB (7KK5) | 7KK5 | ||
| D0120 | Toll-like receptor 7 | Q9NYK1 | TLR7_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (7CYN) | 7CYN | ||
| D0121 | Protein kinase C theta | Q04759 | KPCT_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (5F9E) | 5F9E | ||
| D0122 | P2Y purinoceptor 12 | Q9H244 | P2Y12_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (4TNJ) | 4TNJ | ||
| D0123 | Rotamase A | P62937 | PPIA_HUMAN | chaperone | Successful | Downloaded from PDB (4N1M) | 4N1M | ||
| D0124 | Voltage-gated calcium channel alpha Cav1.3 | Q01668 | CAC1D_HUMAN | voltage-gated ion channel | Clinical trial | Downloaded from PDB (8E59) | 8E59 | ||
| D0125 | Fibroblast growth factor receptor 1 | P11362 | FGFR1_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5EW8) | 5EW8 | ||
| D0126 | Ileal sodium/bile acid cotransporter | Q12908 | NTCP2_HUMAN | primary active transporter | Successful | Modelled with SWISS-MODEL (7PQG.1.B) | HOMOLOGY | ||
| D0127 | Nuclear receptor ROR-gamma | P51449 | RORG_HUMAN | C4 zinc finger nuclear receptor | Clinical trial | Downloaded from PDB (6W9I) | 6W9I | ||
| D0128 | Free fatty acid receptor 1 | O14842 | FFAR1_HUMAN | Undefined | Clinical trial | Downloaded from PDB (5TZR) | 5TZR | ||
| D0129 | Opioid receptor mu | P35372 | OPRM_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (8EFO) | 8EFO | ||
| D0130 | Insulin-like growth factor I receptor | P08069 | IGF1R_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (3LW0) | 3LW0 | ||
| D0131 | RAC-beta serine/threonine-protein kinase | P31751 | AKT2_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (2X39) | 2X39 | ||
| D0132 | Histone acetyltransferase p300 | Q09472 | EP300_HUMAN | histone modifying enzyme | Clinical trial | Downloaded from PDB (5LPM) | 5LPM | ||
| D0133 | Cytochrome P450 2A6 | P11509 | CP2A6_HUMAN | oxygenase | Successful | Downloaded from PDB (2FDV) | 2FDV | ||
| D0134 | Glycoprotein IIb/IIIa receptor | P08514+P05106 | ITA2B_HUMAN+ITB3_HUMAN | integrin | Successful | Downloaded from PDB (7UDH) | 7UDH | ||
| D0135 | Histamine H4 receptor | Q9H3N8 | HRH4_HUMAN | G-protein coupled receptor | Clinical trial | Modelled with SWISS-MODEL (7F61.1.A) | HOMOLOGY | ||
| D0136 | Voltage-gated calcium channel alpha Cav1.2 | Q13936 | CAC1C_HUMAN | voltage-gated ion channel | Successful | Modelled with SWISS-MODEL (7UHG.1.B) | HOMOLOGY | ||
| D0137 | Rho-associated protein kinase 1 | Q13464 | ROCK1_HUMAN | non-receptor serine/threonine protein kinase | Successful | Downloaded from PDB (3V8S) | 3V8S | ||
| D0138 | Adrenergic receptor beta-3 | P13945 | ADRB3_HUMAN | G-protein coupled receptor | Successful | Modelled with SWISS-MODEL (7DH5.1.E) | HOMOLOGY | ||
| D0139 | C-X-C chemokine receptor type 1 | P25024 | CXCR1_HUMAN | cell adhesion molecule | Successful | Modelled with SWISS-MODEL (6LFO.1.E) | HOMOLOGY | ||
| D0140 | Carbonic anhydrase VI | P23280 | CAH6_HUMAN | dehydratase | Successful | Downloaded from PDB (3FE4) | 3FE4 | ||
| D0141 | Farnesoid X-activated receptor | Q96RI1 | NR1H4_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (6HL1) | 6HL1 | ||
| D0142 | GABA A receptor alpha-2 | P47869 | GBRA2_HUMAN | ligand-gated ion channel | Successful | Modelled with SWISS-MODEL (6HUO.1.A) | HOMOLOGY | ||
| D0143 | GABA A receptor alpha-1 | P14867 | GBRA1_HUMAN | ligand-gated ion channel | Successful | Downloaded from PDB (6X3T) | 6X3T | ||
| D0144 | Gastric H+/K+ ATPase alpha | P20648 | ATP4A_HUMAN | primary active transporter | Successful | Modelled with SWISS-MODEL (5YLV.1.A) | HOMOLOGY | ||
| D0145 | Cholecystokinin receptor type A | P32238 | CCKAR_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (7F8Y) | 7F8Y | ||
| D0146 | Matrix metalloproteinase-1 | P03956 | MMP1_HUMAN | metalloprotease | Successful | Downloaded from PDB (966C) | 966C | ||
| D0147 | Kinesin-like protein KIF11 | P52732 | KIF11_HUMAN | microtubule binding motor protein | Clinical trial | Downloaded from PDB (6G6Y) | 6G6Y | ||
| D0148 | Serine/threonine-protein kinase Chk2 | O96017 | CHK2_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (2YCF) | 2YCF | ||
| D0149 | Adrenergic receptor beta-2 | P07550 | ADRB2_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6PS2) | 6PS2 | ||
| D0150 | Histone deacetylase 8 | Q9BY41 | HDAC8_HUMAN | Undefined | Clinical trial | Downloaded from PDB (5VI6) | 5VI6 | ||
| D0151 | Carbonic anhydrase IV | P22748 | CAH4_HUMAN | dehydratase | Successful | Downloaded from PDB (3FW3) | 3FW3 | ||
| D0152 | Platelet-derived growth factor receptor alpha | P16234 | PGFRA_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5GRN) | 5GRN | ||
| D0153 | Neuromedin-K receptor | P29371 | NK3R_HUMAN | G-protein coupled receptor | Successful | Modelled with AlphaFold (AF-P29371-F1-model_v4) | AB INITIO | ||
| D0154 | cAMP-dependent chloride channel F508 deletion | P13569 | CFTR_HUMAN | ATP-binding cassette (ABC) transporter | Successful | Downloaded from PDB (5TFJ) | 5TFJ | ||
| D0155 | Dopamine transporter | Q01959 | SC6A3_HUMAN | primary active transporter | Successful | Modelled with SWISS-MODEL (6VRH.1.A) | HOMOLOGY | ||
| D0156 | Prostaglandin E synthase | O14684 | PTGES_HUMAN | transferase | Clinical trial | Downloaded from PDB (5TL9) | 5TL9 | ||
| D0157 | C-C chemokine receptor type 4 | P51679 | CCR4_HUMAN | cell adhesion molecule | Successful | Modelled with SWISS-MODEL (7O7F.1.C) | HOMOLOGY | ||
| D0158 | ALK tyrosine kinase receptor | Q9UM73 | ALK_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (4Z55) | 4Z55 | ||
| D0159 | ATP-binding cassette transporter G2 | Q9UNQ0 | ABCG2_HUMAN | ATP-binding cassette (ABC) transporter | Successful | Downloaded from PDB (6ETI) | 6ETI | ||
| D0160 | C-X-C chemokine receptor type 2 | P25025 | CXCR2_HUMAN | cell adhesion molecule | Successful | Downloaded from PDB (6LFO) | 6LFO | ||
| D0161 | Debrisoquine 4-hydroxylase | P10635 | CP2D6_HUMAN | oxygenase | Successful | Downloaded from PDB (3TBG) | 3TBG | ||
| D0162 | Lysosomal alpha-glucosidase | P10253 | LYAG_HUMAN | glucosidase | Successful | Downloaded from PDB (5NN5) | 5NN5 | ||
| D0163 | Tyrosine-protein kinase Kit | P10721 | KIT_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (3G0E) | 3G0E | ||
| D0164 | Peroxisome proliferator-activated receptor gamma | P37231 | PPARG_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (2Q59) | 2Q59 | ||
| D0165 | Opioid receptor delta | P41143 | OPRD_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6PT3) | 6PT3 | ||
| D0166 | Platelet-derived growth factor receptor beta | P09619 | PGFRB_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (3MJG) | 3MJG | ||
| D0167 | Sphingosine kinase 2 | Q9NRA0 | SPHK2_HUMAN | kinase | Clinical trial | Modelled with AlphaFold (AF-Q9NRA0-F1-model_v4) | AB INITIO | ||
| D0168 | Epidermal growth factor receptor | P00533 | EGFR_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (8A27) | 8A27 | ||
| D0169 | D-amino acid oxidase | P14920 | OXDA_HUMAN | oxidase | Clinical trial | Downloaded from PDB (7U9U) | 7U9U | ||
| D0170 | Glucagon receptor | P47871 | GLR_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5EE7) | 5EE7 | ||
| D0171 | Prostaglandin G/H synthase 1 | P23219 | PGH1_HUMAN | oxygenase | Successful | Downloaded from PDB (6Y3C) | 6Y3C | ||
| D0172 | Tropomyosin-related kinase A | P04629 | NTRK1_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5JFW) | 5JFW | ||
| D0173 | Thyrotropin receptor | P16473 | TSHR_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7T9M) | 7T9M | ||
| D0174 | Proto-oncogene c-Ret | P07949 | RET_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (7DUA) | 7DUA | ||
| D0175 | Opioid receptor kappa | P41145 | OPRK_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (8DZR) | 8DZR | ||
| D0176 | Matrix metalloproteinase-13 | P45452 | MMP13_HUMAN | metalloprotease | Clinical trial | Downloaded from PDB (3ZXH) | 3ZXH | ||
| D0177 | Dihydrodiol dehydrogenase type I | P42330 | AK1C3_HUMAN | reductase | Successful | Downloaded from PDB (1S1P) | 1S1P | ||
| D0178 | Dihydroorotate dehydrogenase | Q02127 | PYRD_HUMAN | dehydrogenase | Successful | Downloaded from PDB (4OQV) | 4OQV | ||
| D0179 | Angiotensinogenase renin | P00797 | RENI_HUMAN | aspartic protease | Successful | Downloaded from PDB (3K1W) | 3K1W | ||
| D0180 | Phosphodiesterase 4A | P27815 | PDE4A_HUMAN | phosphodiesterase | Successful | Downloaded from PDB (2QYK) | 2QYK | ||
| D0181 | Soluble epoxide hydrolase | P34913 | HYES_HUMAN | hydrolase | Clinical trial | Downloaded from PDB (4JNC) | 4JNC | ||
| D0182 | ERK activator kinase 1 | Q02750 | MP2K1_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (7B7R) | 7B7R | ||
| D0183 | Adenosine A3 receptor | P0DMS8 | AA3R_HUMAN | G-protein coupled receptor | Clinical trial | Modelled with SWISS-MODEL (7LD3.1.B) | HOMOLOGY | ||
| D0184 | Glutamate receptor ionotropic NMDA 1 | Q05586 | NMDZ1_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5H8Q) | 5H8Q | ||
| D0185 | GABA A receptor alpha-3 | P34903 | GBRA3_HUMAN | ligand-gated ion channel | Successful | Modelled with SWISS-MODEL (6HUG.1.A) | HOMOLOGY | ||
| D0186 | Peroxisome proliferator-activated receptor delta | Q03181 | PPARD_HUMAN | C4 zinc finger nuclear receptor | Clinical trial | Downloaded from PDB (5Y7X) | 5Y7X | ||
| D0187 | Tyrosine-protein kinase SYK | P43405 | KSYK_HUMAN | non-receptor tyrosine protein kinase | Successful | Downloaded from PDB (4YJR) | 4YJR | ||
| D0188 | Bacterial Dihydrofolate reductase | P0ABQ4 | DYR_ECOLI | reductase | Clinical trial | Downloaded from PDB (6MT8) | 6MT8 | ||
| D0189 | Vascular endothelial growth factor receptor 3 | P35916 | VGFR3_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (4BSJ) | 4BSJ | ||
| D0190 | Janus kinase 1 | P23458 | JAK1_HUMAN | non-receptor tyrosine protein kinase | Successful | Downloaded from PDB (6N7A) | 6N7A | ||
| D0191 | Tyrosine-protein kinase ABL1 | P00519 | ABL1_HUMAN | non-receptor tyrosine protein kinase | Successful | Downloaded from PDB (5HU9) | 5HU9 | ||
| D0192 | Cathepsin A | P10619 | PPGB_HUMAN | serine protease | Clinical trial | Downloaded from PDB (4CIB) | 4CIB | ||
| D0193 | Vascular endothelial growth factor receptor 1 | P17948 | VGFR1_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (3HNG) | 3HNG | ||
| D0194 | Nitric-oxide synthase inducible | P35228 | NOS2_HUMAN | oxidoreductase | Clinical trial | Downloaded from PDB (3E7G) | 3E7G | ||
| D0195 | Neuronal acetylcholine receptor alpha-4/beta-2 | P43681+P17787 | ACHA4_HUMAN+ACHB2_HUMAN | ligand-gated ion channel | Successful | Downloaded from PDB (5KXI) | 5KXI | ||
| D0196 | Albendazole monooxygenase | P08684 | CP3A4_HUMAN | oxygenase | Clinical trial | Downloaded from PDB (4D6Z) | 4D6Z | ||
| D0197 | 5-HT 3A receptor | P46098 | 5HT3A_HUMAN | ligand-gated ion channel | Successful | Modelled with SWISS-MODEL (6NP0.1.A) | HOMOLOGY | ||
| D0198 | Histamine H3 receptor | Q9Y5N1 | HRH3_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7F61) | 7F61 | ||
| D0199 | Voltage-gated calcium channel alpha Cav3.1 | O43497 | CAC1G_HUMAN | voltage-gated ion channel | Successful | Downloaded from PDB (6KZP) | 6KZP | ||
| D0200 | Somatostatin receptor type 5 | P35346 | SSR5_HUMAN | G-protein coupled receptor | Successful | Modelled with SWISS-MODEL (7UL5.1.A) | HOMOLOGY | ||
| D0201 | Ubiquitin-protein ligase E3 Mdm2 | Q00987 | MDM2_HUMAN | Undefined | Clinical trial | Downloaded from PDB (6Q96) | 6Q96 | ||
| D0202 | Coagulation factor XII | P00748 | FA12_HUMAN | serine protease | Clinical trial | Downloaded from PDB (6X0T) | 6X0T | ||
| D0203 | dUTP pyrophosphatase | P33316 | DUT_HUMAN | phosphatase | Clinical trial | Downloaded from PDB (3ARA) | 3ARA | ||
| D0204 | Ras-related protein Rab-9A | P51151 | RAB9A_HUMAN | small GTPase | Successful | Downloaded from PDB (1WMS) | 1WMS | ||
| D0205 | Smoothened homolog | Q99835 | SMO_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (7ZI0) | 7ZI0 | ||
| D0206 | Prostaglandin G/H synthase 2 | P35354 | PGH2_HUMAN | oxygenase | Successful | Downloaded from PDB (5F1A) | 5F1A | ||
| D0207 | Dopamine D2 receptor | P14416 | DRD2_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6CM4) | 6CM4 | ||
| D0208 | Neurotensin receptor type 1 | P30989 | NTR1_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (7UL2) | 7UL2 | ||
| D0209 | Macrophage migration inhibitory factor | P14174 | MIF_HUMAN | decarboxylase | Clinical trial | Downloaded from PDB (6B1K) | 6B1K | ||
| D0210 | Muscarinic acetylcholine receptor M3 | P20309 | ACM3_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (8EA0) | 8EA0 | ||
| D0211 | PI3-kinase delta | O00329 | PK3CD_HUMAN | kinase | Successful | Downloaded from PDB (6PYR) | 6PYR | ||
| D0212 | Stress-activated protein kinase JNK1 | P45983 | MK08_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (3ELJ) | 3ELJ | ||
| D0213 | DNA-binding factor KBF1 | P19838 | NFKB1_HUMAN | Rel homology transcription factor | Clinical trial | Downloaded from PDB (1SVC) | 1SVC | ||
| D0214 | Protein kinase C beta | P05771 | KPCB_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (2I0E) | 2I0E | ||
| D0215 | Matrix metalloproteinase-2 | P08253 | MMP2_HUMAN | metalloprotease | Successful | Downloaded from PDB (7XJO) | 7XJO | ||
| D0216 | Neutrophil elastase | P08246 | ELNE_HUMAN | serine protease | Clinical trial | Downloaded from PDB (5ABW) | 5ABW | ||
| D0217 | Follicle-stimulating hormone receptor | P23945 | FSHR_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (8I2G) | 8I2G | ||
| D0218 | Bromodomain-containing protein 4 | O60885 | BRD4_HUMAN | Undefined | Clinical trial | Downloaded from PDB (6FO5) | 6FO5 | ||
| D0219 | Histone deacetylase 1 | Q13547 | HDAC1_HUMAN | Undefined | Successful | Downloaded from PDB (4BKX) | 4BKX | ||
| D0220 | Polo-like kinase 1 | P53350 | PLK1_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (4X9R) | 4X9R | ||
| D0221 | Phosphodiesterase 5A | O76074 | PDE5A_HUMAN | phosphodiesterase | Successful | Downloaded from PDB (2H44) | 2H44 | ||
| D0222 | Orexin receptor type 2 | O43614 | OX2R_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7L1V) | 7L1V | ||
| D0223 | Cathepsin L | P07711 | CATL1_HUMAN | cysteine protease | Clinical trial | Downloaded from PDB (2XU3) | 2XU3 | ||
| D0224 | Survival motor neuron protein | Q16637 | SMN_HUMAN | RNA splicing factor | Successful | Downloaded from PDB (7W2P) | 7W2P | ||
| D0225 | Melanocortin receptor 4 | P32245 | MC4R_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7PIU) | 7PIU | ||
| D0226 | Leukocyte common antigen | P08575 | PTPRC_HUMAN | protein phosphatase | Clinical trial | Downloaded from PDB (1YGU) | 1YGU | ||
| D0227 | Matrix metalloproteinase-7 | P09237 | MMP7_HUMAN | metalloprotease | Successful | Downloaded from PDB (1MMQ) | 1MMQ | ||
| D0228 | Estradiol 17 beta-dehydrogenase 1 | P14061 | DHB1_HUMAN | dehydrogenase | Clinical trial | Downloaded from PDB (1JTV) | 1JTV | ||
| D0229 | Glutamate receptor ionotropic kainate 1 | P39086 | GRIK1_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (3FV1) | 3FV1 | ||
| D0230 | Cyclin-dependent kinase 9 | P50750 | CDK9_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (3BLR) | 3BLR | ||
| D0231 | Neuronal acetylcholine receptor alpha-3/beta-4 | P32297+P30926 | ACHA3_HUMAN-ACHB4_HUMAN | ligand-gated ion channel | Successful | Downloaded from PDB (6PV7) | 6PV7 | ||
| D0232 | Fms-like tyrosine kinase 3 | P36888 | FLT3_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (6JQR) | 6JQR | ||
| D0233 | Angiotensin II receptor type-1 | P30556 | AGTR1_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6OS2) | 6OS2 | ||
| D0234 | Serine/threonine-protein kinase mTOR | P42345 | MTOR_HUMAN | non-receptor serine/threonine protein kinase | Successful | Modelled with SWISS-MODEL (6ZWM.1.A) | HOMOLOGY | ||
| D0235 | Tryptophan 2,3-dioxygenase | P48775 | T23O_HUMAN | oxygenase | Clinical trial | Downloaded from PDB (6PYZ) | 6PYZ | ||
| D0236 | Janus kinase 2 | O60674 | JAK2_HUMAN | non-receptor tyrosine protein kinase | Successful | Downloaded from PDB (7LL4) | 7LL4 | ||
| D0237 | Staphylococcus DNA gyrase A | P20831 | GYRA_STAAU | Undefined | Successful | Downloaded from PDB (7MVS) | 7MVS | ||
| D0238 | Protein kinase C delta | Q05655 | KPCD_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Modelled with SWISS-MODEL (3PFQ.1.A) | HOMOLOGY | ||
| D0239 | Quinone reductase 2 | P16083 | NQO2_HUMAN | oxidoreductase | Successful | Downloaded from PDB (4FGL) | 4FGL | ||
| D0240 | Carnitine O-palmitoyltransferase I | Q92523 | CPT1B_HUMAN | acyltransferase | Successful | Modelled with AlphaFold (AF-Q92523-F1-model_v4) | AB INITIO | ||
| D0241 | FK506-binding protein 1A | P62942 | FKB1A_HUMAN | chaperone | Successful | Downloaded from PDB (6YF3) | 6YF3 | ||
| D0242 | Thromboxane A2 receptor | P21731 | TA2R_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6IIU) | 6IIU | ||
| D0243 | Liver carboxylesterase | P23141 | EST1_HUMAN | esterase | Successful | Downloaded from PDB (5A7F) | 5A7F | ||
| D0244 | Glutamate receptor ionotropic NMDA 2B | Q13224 | NMDE2_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5EWM) | 5EWM | ||
| D0245 | Coagulation factor XI | P03951 | FA11_HUMAN | serine protease | Clinical trial | Downloaded from PDB (6TS4) | 6TS4 | ||
| D0246 | Cannabinoid receptor 1 | P21554 | CNR1_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (5XRA) | 5XRA | ||
| D0247 | Glycogen synthase kinase-3 alpha | P49840 | GSK3A_HUMAN | non-receptor serine/threonine protein kinase | Successful | Modelled with SWISS-MODEL (6AE3.1.A) | HOMOLOGY | ||
| D0248 | Glutaminyl cyclase | Q16769 | QPCT_HUMAN | transferase | Clinical trial | Downloaded from PDB (2AFX) | 2AFX | ||
| D0249 | M-phase inducer phosphatase 2 | P30305 | MPIP2_HUMAN | protein phosphatase | Clinical trial | Downloaded from PDB (4WH9) | 4WH9 | ||
| D0250 | Matrix metalloproteinase-12 | P39900 | MMP12_HUMAN | metalloprotease | Clinical trial | Downloaded from PDB (6EKN) | 6EKN | ||
| D0251 | Adenosine A2a receptor | P29274 | AA2AR_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (3VG9) | 3VG9 | ||
| D0252 | Bacterial Botulinum toxin A | P0DPI0 | BXA1_CLOBO | Undefined | Clinical trial | Downloaded from PDB (6XCF) | 6XCF | ||
| D0253 | Histamine H1 receptor | P35367 | HRH1_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7DFL) | 7DFL | ||
| D0254 | Aurora kinase B | Q96GD4 | AURKB_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (4AF3) | 4AF3 | ||
| D0255 | 5-HT 1A receptor | P08908 | 5HT1A_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7E2Y) | 7E2Y | ||
| D0256 | Bacterial Fatty acid synthetase I | P9WGR1 | INHA_MYCTU | reductase | Successful | Downloaded from PDB (4OHU) | 4OHU | ||
| D0257 | Thyroid hormone receptor alpha | P10827 | THA_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (3HZF) | 3HZF | ||
| D0258 | Muscarinic acetylcholine receptor M5 | P08912 | ACM5_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6OL9) | 6OL9 | ||
| D0259 | PI3-kinase alpha | P42336 | PK3CA_HUMAN | kinase | Successful | Downloaded from PDB (8EXL) | 8EXL | ||
| D0260 | GABA A receptor beta-2 | P47870 | GBRB2_HUMAN | ligand-gated ion channel | Successful | Downloaded from PDB (6X3T) | 6X3T | ||
| D0261 | Toll-like receptor 8 | Q9NR97 | TLR8_HUMAN | transmembrane signal receptor | Clinical trial | Downloaded from PDB (3WN4) | 3WN4 | ||
| D0262 | Estrogen receptor beta | Q92731 | ESR2_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (1QKM) | 1QKM | ||
| D0263 | Urotensin II receptor | Q9UKP6 | UR2R_HUMAN | G-protein coupled receptor | Clinical trial | Modelled with AlphaFold (AF-Q9UKP6-F1-model_v4) | AB INITIO | ||
| D0264 | Acetyl-CoA carboxylase 2 | O00763 | ACACB_HUMAN | Undefined | Successful | Downloaded from PDB (3GID) | 3GID | ||
| D0265 | Vascular endothelial growth factor receptor 2 | P35968 | VGFR2_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (3VHE) | 3VHE | ||
| D0266 | Tyrosine-protein phosphatase non-receptor type 2 | P17706 | PTN2_HUMAN | protein phosphatase | Clinical trial | Downloaded from PDB (7F5O) | 7F5O | ||
| D0267 | Tyrosine-protein kinase UFO | P30530 | UFO_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5U6B) | 5U6B | ||
| D0268 | Angiotensin-converting enzyme | P12821 | ACE_HUMAN | metalloprotease | Successful | Downloaded from PDB (6F9T) | 6F9T | ||
| D0269 | Ephrin type-B receptor 4 | P54760 | EPHB4_HUMAN | transmembrane signal receptor | Clinical trial | Downloaded from PDB (6FNM) | 6FNM | ||
| D0270 | Plasma kallikrein | P03952 | KLKB1_HUMAN | serine protease | Successful | Downloaded from PDB (6O1S) | 6O1S | ||
| D0271 | Cyclin-dependent kinase 1 | P06493 | CDK1_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (4Y72) | 4Y72 | ||
| D0272 | CREB-binding protein | Q92793 | CBP_HUMAN | histone modifying enzyme | Clinical trial | Downloaded from PDB (5I86) | 5I86 | ||
| D0273 | Monoamine oxidase type B | P27338 | AOFB_HUMAN | oxidase | Successful | Downloaded from PDB (2XCG) | 2XCG | ||
| D0274 | TGF-beta receptor type II | P37173 | TGFR2_HUMAN | serine/threonine protein kinase receptor | Clinical trial | Downloaded from PDB (4XJJ) | 4XJJ | ||
| D0275 | Sphingosine-1-phosphate receptor 5 | Q9H228 | S1PR5_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (7YXA) | 7YXA | ||
| D0276 | Transient receptor potential cation channel V1 | Q8NER1 | TRPV1_HUMAN | ion channel | Successful | Downloaded from PDB (8GFA) | 8GFA | ||
| D0277 | Serine/threonine-protein kinase pim-1 | P11309 | PIM1_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (3R04) | 3R04 | ||
| D0278 | 5-HT 2C receptor | P28335 | 5HT2C_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6BQH) | 6BQH | ||
| D0279 | Monoamine oxidase type A | P21397 | AOFA_HUMAN | oxidase | Successful | Downloaded from PDB (2Z5X) | 2Z5X | ||
| D0280 | Transformation-sensitive protein p120 | O75762 | TRPA1_HUMAN | scaffold/adaptor protein | Successful | Downloaded from PDB (6PQO) | 6PQO | ||
| D0281 | Histone deacetylase 2 | Q92769 | HDAC2_HUMAN | Undefined | Clinical trial | Downloaded from PDB (7KBG) | 7KBG | ||
| D0282 | Steroid 11-beta-hydroxylase | P15538 | C11B1_HUMAN | Undefined | Successful | Downloaded from PDB (6M7X) | 6M7X | ||
| D0283 | Coagulation factor Xa | P00742 | FA10_HUMAN | serine protease | Successful | Downloaded from PDB (2JKH) | 2JKH | ||
| D0284 | Casein kinase II alpha | P68400 | CSK21_HUMAN | Undefined | Clinical trial | Downloaded from PDB (8AEC) | 8AEC | ||
| D0285 | BDNF/NT-3 growth factors receptor | Q16620 | NTRK2_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (4AT5) | 4AT5 | ||
| D0286 | Insulin receptor | P06213 | INSR_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (5HHW) | 5HHW | ||
| D0287 | Cyclin-dependent kinase 4 | P11802 | CDK4_HUMAN | non-receptor serine/threonine protein kinase | Successful | Downloaded from PDB (7SJ3) | 7SJ3 | ||
| D0288 | Proto-oncogene c-Src | P12931 | SRC_HUMAN | non-receptor tyrosine protein kinase | Successful | Downloaded from PDB (1O43) | 1O43 | ||
| D0289 | Geranyltranstransferase | P14324 | FPPS_HUMAN | acyltransferase | Successful | Downloaded from PDB (5CG5) | 5CG5 | ||
| D0290 | Peroxisome proliferator-activated receptor alpha | Q07869 | PPARA_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (1i7g) | 1i7g | ||
| D0291 | Alkaline phosphatase tissue-nonspecific | P05186 | PPBT_HUMAN | phosphatase | Successful | Modelled with SWISS-MODEL (4KJD.1.A) | HOMOLOGY | ||
| D0292 | Substance-K receptor | P21452 | NK2R_HUMAN | G-protein coupled receptor | Clinical trial | Modelled with SWISS-MODEL (7MRG.1.B) | HOMOLOGY | ||
| D0293 | Adenosine A2b receptor | P29275 | AA2BR_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (8HDO) | 8HDO | ||
| D0294 | Amyloid beta A4 protein | P05067 | A4_HUMAN | protease inhibitor | Successful | Modelled with AlphaFold (AF-P05067-F1-model_v4) | AB INITIO | ||
| D0295 | TGF-beta receptor type I | P36897 | TGFR1_HUMAN | serine/threonine protein kinase receptor | Clinical trial | Downloaded from PDB (4X2F) | 4X2F | ||
| D0296 | G-protein coupled receptor 55 | Q9Y2T6 | GPR55_HUMAN | G-protein coupled receptor | Successful | Modelled with SWISS-MODEL (7F2O.1.C) | HOMOLOGY | ||
| D0297 | Prolyl endopeptidase FAP | Q12884 | SEPR_HUMAN | serine protease | Clinical trial | Downloaded from PDB (6Y0F) | 6Y0F | ||
| D0298 | Nicotinic acid receptor | Q8TDS4 | HCAR2_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7XK2) | 7XK2 | ||
| D0299 | HIF-prolyl hydroxylase 1 | Q96KS0 | EGLN2_HUMAN | Undefined | Successful | Downloaded from PDB (5V1B) | 5V1B | ||
| D0300 | DNA topoisomerase I | P11387 | TOP1_HUMAN | DNA topoisomerase | Successful | Downloaded from PDB (1A36) | 1A36 | ||
| D0301 | Phosphodiesterase 3A | Q14432 | PDE3A_HUMAN | phosphodiesterase | Successful | Downloaded from PDB (7KWE) | 7KWE | ||
| D0302 | Plasminogen | P00747 | PLMN_HUMAN | serine protease | Successful | Downloaded from PDB (5UGG) | 5UGG | ||
| D0303 | Matrix metalloproteinase-9 | P14780 | MMP9_HUMAN | metalloprotease | Clinical trial | Downloaded from PDB (6ESM) | 6ESM | ||
| D0304 | Nicotinamide phosphoribosyltransferase | P43490 | NAMPT_HUMAN | transferase | Clinical trial | Downloaded from PDB (6E68) | 6E68 | ||
| D0305 | Estrogen receptor | P03372 | ESR1_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (7UJO) | 7UJO | ||
| D0306 | Sodium/glucose cotransporter 1 | P13866 | SC5A1_HUMAN | secondary carrier transporter | Clinical trial | Downloaded from PDB (7WMV) | 7WMV | ||
| D0307 | Indoleamine 2,3-dioxygenase 1 | P14902 | I23O1_HUMAN | oxygenase | Successful | Downloaded from PDB (8ABX) | 8ABX | ||
| D0308 | Erbb4 tyrosine kinase receptor | Q15303 | ERBB4_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (2R4B) | 2R4B | ||
| D0309 | Adenosine A1 receptor | P30542 | AA1R_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (5UEN) | 5UEN | ||
| D0310 | Renal carcinoma antigen NY-REN-64 | Q9NWZ3 | IRAK4_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (6EGE) | 6EGE | ||
| D0311 | Hypoxia-inducible factor 1 alpha | Q16665 | HIF1A_HUMAN | basic helix-loop-helix transcription factor | Clinical trial | Downloaded from PDB (4H6J) | 4H6J | ||
| D0312 | Choline kinase | P35790 | CHKA_HUMAN | kinase | Clinical trial | Downloaded from PDB (5FTG) | 5FTG | ||
| D0313 | Stress-activated protein kinase 2b | Q15759 | MK11_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (3GP0) | 3GP0 | ||
| D0314 | C-C chemokine receptor type 5 | P51681 | CCR5_HUMAN | cell adhesion molecule | Successful | Downloaded from PDB (6AKX) | 6AKX | ||
| D0315 | Tyrosine-protein kinase Mer | Q12866 | MERTK_HUMAN | transmembrane signal receptor | Clinical trial | Downloaded from PDB (7AAZ) | 7AAZ | ||
| D0316 | Intestinal maltase-glucoamylase | O43451 | MGA_HUMAN | glucosidase | Successful | Downloaded from PDB (3L4Y) | 3L4Y | ||
| D0317 | Endothelin B receptor | P24530 | EDNRB_HUMAN | Undefined | Successful | Downloaded from PDB (6IGK) | 6IGK | ||
| D0318 | Apoptosis regulator Bcl-xL | Q07817 | B2CL1_HUMAN | Undefined | Clinical trial | Downloaded from PDB (7LH7) | 7LH7 | ||
| D0319 | Coagulation factor IIa | P00734 | THRB_HUMAN | serine protease | Successful | Downloaded from PDB (5AFY) | 5AFY | ||
| D0320 | Ephrin type-A receptor 2 | P29317 | EPHA2_HUMAN | transmembrane signal receptor | Clinical trial | Downloaded from PDB (6HET) | 6HET | ||
| D0321 | Caspase-3 | P42574 | CASP3_HUMAN | protease | Clinical trial | Downloaded from PDB (6X8I) | 6X8I | ||
| D0322 | PI3-kinase gamma | P48736 | PK3CG_HUMAN | kinase | Successful | Downloaded from PDB (4ANV) | 4ANV | ||
| D0323 | Cyclin-dependent kinase 7 | P50613 | CDK7_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (7B5Q) | 7B5Q | ||
| D0324 | C-X-C chemokine receptor type 4 | P61073 | CXCR4_HUMAN | cell adhesion molecule | Successful | Downloaded from PDB (3ODU) | 3ODU | ||
| D0325 | Transient receptor potential cation channel V3 | Q8NET8 | TRPV3_HUMAN | ion channel | Clinical trial | Downloaded from PDB (6UW4) | 6UW4 | ||
| D0326 | B1 bradykinin receptor | P46663 | BKRB1_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (7EIB) | 7EIB | ||
| D0327 | Voltage-gated sodium channel alpha Nav1.6 | Q9UQD0 | SCN8A_HUMAN | voltage-gated ion channel | Clinical trial | Downloaded from PDB (8FHD) | 8FHD | ||
| D0328 | Beta-glucuronidase | P08236 | BGLR_HUMAN | Undefined | Successful | Downloaded from PDB (3HN3) | 3HN3 | ||
| D0329 | Extracellular signal-regulated kinase 2 | P28482 | MK01_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (4ZZN) | 4ZZN | ||
| D0330 | Acyl-CoA desaturase | O00767 | SCD_HUMAN | Undefined | Successful | Downloaded from PDB (4ZYO) | 4ZYO | ||
| D0331 | Thyroid hormone receptor beta | P10828 | THB_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (2J4A) | 2J4A | ||
| D0332 | Serine/threonine-protein kinase B-raf | P15056 | BRAF_HUMAN | non-receptor serine/threonine protein kinase | Successful | Downloaded from PDB (8C7Y) | 8C7Y | ||
| D0333 | Trace amine-associated receptor-1 | Q96RJ0 | TAAR1_HUMAN | G-protein coupled receptor | Successful | Modelled with SWISS-MODEL (7CKY.1.E) | HOMOLOGY | ||
| D0334 | PI3-kinase beta | P42338 | PK3CB_HUMAN | kinase | Clinical trial | Modelled with SWISS-MODEL (2Y3A.1.A) | HOMOLOGY | ||
| D0335 | Prostaglandin D2 receptor 2 | Q9Y5Y4 | PD2R2_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (6D26) | 6D26 | ||
| D0336 | Checkpoint kinase-1 | O14757 | CHK1_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (4HYI) | 4HYI | ||
| D0337 | Histone deacetylase 3 | O15379 | HDAC3_HUMAN | Undefined | Clinical trial | Downloaded from PDB (4A69) | 4A69 | ||
| D0338 | P2X purinoceptor 7 | Q99572 | P2RX7_HUMAN | ligand-gated ion channel | Clinical trial | Modelled with SWISS-MODEL (6U9W.1.A) | HOMOLOGY | ||
| D0339 | Histone deacetylase 4 | P56524 | HDAC4_HUMAN | Undefined | Clinical trial | Downloaded from PDB (2VQM) | 2VQM | ||
| D0340 | Androgen receptor | P10275 | ANDR_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (2AM9) | 2AM9 | ||
| D0341 | Chymase | P23946 | CMA1_HUMAN | serine protease | Clinical trial | Downloaded from PDB (4K69) | 4K69 | ||
| D0342 | Carbonic anhydrase IX | Q16790 | CAH9_HUMAN | dehydratase | Clinical trial | Downloaded from PDB (6G9U) | 6G9U | ||
| D0343 | Matrix metalloproteinase-14 | P50281 | MMP14_HUMAN | metalloprotease | Clinical trial | Downloaded from PDB (3MA2) | 3MA2 | ||
| D0344 | Multidrug resistance-associated protein 1 | P33527 | MRP1_HUMAN | ATP-binding cassette (ABC) transporter | Successful | Downloaded from PDB (2CBZ) | 2CBZ | ||
| D0345 | Corticosteroid 11-beta-dehydrogenase 1 | P28845 | DHI1_HUMAN | dehydrogenase | Clinical trial | Downloaded from PDB (4BB5) | 4BB5 | ||
| D0346 | Stress-activated protein kinase 2a | Q16539 | MK14_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (3LFF) | 3LFF | ||
| D0347 | Pyruvate kinase M2 | P14618 | KPYM_HUMAN | kinase | Clinical trial | Downloaded from PDB (8G2E) | 8G2E | ||
| D0348 | Adrenergic receptor alpha-2A | P08913 | ADA2A_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6KUX) | 6KUX | ||
| D0349 | Dipeptidyl peptidase 9 | Q86TI2 | DPP9_HUMAN | serine protease | Clinical trial | Downloaded from PDB (7ZXS) | 7ZXS | ||
| D0350 | Complement factor D | P00746 | CFAD_HUMAN | serine protease | Clinical trial | Downloaded from PDB (5NAT) | 5NAT | ||
| D0351 | Cathepsin D | P07339 | CATD_HUMAN | aspartic protease | Clinical trial | Downloaded from PDB (6QCB) | 6QCB | ||
| D0352 | Aminopeptidase N | P15144 | AMPN_HUMAN | metalloprotease | Clinical trial | Downloaded from PDB (4FYT) | 4FYT | ||
| D0353 | Integrin alpha-V/beta-3 | P06756+P05106 | ITAV_HUMAN+ITB3_HUMAN | integrin | Clinical trial | Downloaded from PDB (6MK0) | 6MK0 | ||
| D0354 | RAC-alpha serine/threonine-protein kinase | P31749 | AKT1_HUMAN | non-receptor serine/threonine protein kinase | Successful | Downloaded from PDB (4GV1) | 4GV1 | ||
| D0355 | Cathepsin S | P25774 | CATS_HUMAN | cysteine protease | Clinical trial | Downloaded from PDB (3OVX) | 3OVX | ||
| D0356 | Gonadotropin-releasing hormone receptor | P30968 | GNRHR_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7BR3) | 7BR3 | ||
| D0357 | Glycine transporter GlyT-1 | P48067 | SC6A9_HUMAN | primary active transporter | Clinical trial | Downloaded from PDB (6ZBV) | 6ZBV | ||
| D0358 | Adrenergic receptor alpha-2C | P18825 | ADA2C_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (6KUW) | 6KUW | ||
| D0359 | LCK tyrosine protein kinase | P06239 | LCK_HUMAN | non-receptor tyrosine protein kinase | Successful | Downloaded from PDB (6PDJ) | 6PDJ | ||
| D0360 | Cyclin-dependent kinase 2 | P24941 | CDK2_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (4FKL) | 4FKL | ||
| D0361 | Glycogen synthase kinase-3 beta | P49841 | GSK3B_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (1Q5K) | 1Q5K | ||
| D0362 | Protein kinase C alpha | P17252 | KPCA_HUMAN | non-receptor serine/threonine protein kinase | Successful | Downloaded from PDB (4RA4) | 4RA4 | ||
| D0363 | Nitric-oxide synthase endothelial | P29474 | NOS3_HUMAN | oxidoreductase | Clinical trial | Downloaded from PDB (6PP1) | 6PP1 | ||
| D0364 | Caspase-7 | P55210 | CASP7_HUMAN | protease | Clinical trial | Downloaded from PDB (2QL9) | 2QL9 | ||
| D0365 | Bacterial Lethal factor | P15917 | LEF_BACAN | Undefined | Clinical trial | Downloaded from PDB (4PKW) | 4PKW | ||
| D0366 | Tissue factor | P13726 | TF_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (6R2W) | 6R2W | ||
| D0367 | E-selectin | P16581 | LYAM2_HUMAN | complement component | Clinical trial | Downloaded from PDB (1G1T) | 1G1T | ||
| D0368 | Orexin receptor type 1 | O43613 | OX1R_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (6TOT) | 6TOT | ||
| D0369 | Rho-associated protein kinase 2 | O75116 | ROCK2_HUMAN | non-receptor serine/threonine protein kinase | Successful | Downloaded from PDB (7JNT) | 7JNT | ||
| D0370 | Dual specificity protein kinase TTK | P33981 | TTK_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (4JS8) | 4JS8 | ||
| D0371 | Methionine aminopeptidase 2 | P50579 | MAP2_HUMAN | protease | Clinical trial | Downloaded from PDB (6QEJ) | 6QEJ | ||
| D0372 | Farnesyl protein transferase | P49354+P49356 | FNTA_HUMAN+FNTB_HUMAN | acyltransferase | Successful | Downloaded from PDB (1LD8) | 1LD8 | ||
| D0373 | Pattern recognition receptor NOD2 | Q9HC29 | NOD2_HUMAN | scaffold/adaptor protein | Clinical trial | Modelled with SWISS-MODEL (5IRM.1.A) | HOMOLOGY | ||
| D0374 | Geranylgeranyl transferase I | P53609 | PGTB1_HUMAN | acyltransferase | Clinical trial | Modelled with SWISS-MODEL (1TNU.1.B) | HOMOLOGY | ||
| D0375 | Carbonic anhydrase I | P00915 | CAH1_HUMAN | dehydratase | Successful | Downloaded from PDB (7Q0D) | 7Q0D | ||
| D0376 | Proteasome beta-8 | P28062 | PSB8_HUMAN | protease | Clinical trial | Downloaded from PDB (7AWE) | 7AWE | ||
| D0377 | Phosphodiesterase 2A | O00408 | PDE2A_HUMAN | phosphodiesterase | Clinical trial | Downloaded from PDB (5U00) | 5U00 | ||
| D0378 | Thromboxane-A synthase | P24557 | THAS_HUMAN | isomerase | Clinical trial | Downloaded from PDB (5VCE) | 5VCE | ||
| D0379 | Inhibitor of nuclear factor kappa-B kinase beta | O14920 | IKKB_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (4KIK) | 4KIK | ||
| D0380 | TYK2 tyrosine kinase | P29597 | TYK2_HUMAN | non-receptor tyrosine protein kinase | Successful | Downloaded from PDB (4WOV) | 4WOV | ||
| D0381 | Beta-secretase 1 | P56817 | BACE1_HUMAN | protease | Clinical trial | Downloaded from PDB (7MYI) | 7MYI | ||
| D0382 | 5-HT 7 receptor | P34969 | 5HT7R_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (7XTC) | 7XTC | ||
| D0383 | Aromatase | P11511 | CP19A_HUMAN | oxygenase | Successful | Downloaded from PDB (5JKV) | 5JKV | ||
| D0384 | DNA-dependent protein kinase catalytic | P78527 | PRKDC_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Modelled with SWISS-MODEL (7OTV.1.A) | HOMOLOGY | ||
| D0385 | Phosphodiesterase 4D | Q08499 | PDE4D_HUMAN | phosphodiesterase | Successful | Downloaded from PDB (5WH6) | 5WH6 | ||
| D0386 | TNF alpha converting enzyme | P78536 | ADA17_HUMAN | protease | Clinical trial | Downloaded from PDB (2DDF) | 2DDF | ||
| D0387 | Retinoic acid receptor RXR-alpha | P19793 | RXRA_HUMAN | C4 zinc finger nuclear receptor | Successful | Downloaded from PDB (7A77) | 7A77 | ||
| D0388 | Cysteines of Keap1 | Q14145 | KEAP1_HUMAN | scaffold/adaptor protein | Clinical trial | Downloaded from PDB (6TYM) | 6TYM | ||
| D0389 | Phosphodiesterase 10A | Q9Y233 | PDE10_HUMAN | phosphodiesterase | Clinical trial | Downloaded from PDB (5C28) | 5C28 | ||
| D0390 | Sphingosine-1-phosphate receptor 1 | P21453 | S1PR1_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (7TD4) | 7TD4 | ||
| D0391 | Tubulin beta-1 chain | Q9H4B7 | TBB1_HUMAN | tubulin | Clinical trial | Modelled with SWISS-MODEL (6TIS.1.B) | HOMOLOGY | ||
| D0392 | Sphingosine kinase 1 | Q9NYA1 | SPHK1_HUMAN | kinase | Clinical trial | Downloaded from PDB (4V24) | 4V24 | ||
| D0393 | Telomerase reverse transcriptase | O14746 | TERT_HUMAN | DNA metabolism protein | Clinical trial | Downloaded from PDB (5UGW) | 5UGW | ||
| D0394 | Prolyl endopeptidase | P48147 | PPCE_HUMAN | serine protease | Clinical trial | Downloaded from PDB (3DDU) | 3DDU | ||
| D0395 | Solute carrier family 40 member 1 | Q9NP59 | S40A1_HUMAN | secondary carrier transporter | Clinical trial | Downloaded from PDB (8DL7) | 8DL7 | ||
| D0396 | G-protein coupled bile acid receptor 1 | Q8TDU6 | GPBAR_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (7CFM) | 7CFM | ||
| D0397 | Serine/threonine-protein kinase pim-2 | Q9P1W9 | PIM2_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (4X7Q) | 4X7Q | ||
| D0398 | Cathepsin G | P08311 | CATG_HUMAN | serine protease | Clinical trial | Downloaded from PDB (1T32) | 1T32 | ||
| D0399 | Bromodomain-containing protein 2 | P25440 | BRD2_HUMAN | Undefined | Clinical trial | Downloaded from PDB (5IG6) | 5IG6 | ||
| D0400 | Glutaminase | O94925+Q9UI32 | GLSK_HUMAN+GLSL_HUMAN | hydrolase | Clinical trial | Downloaded from PDB (8BSK) | 8BSK | ||
| D0401 | Aurora kinase A | O14965 | AURKA_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (5L8L) | 5L8L | ||
| D0402 | N-formyl peptide receptor | P21462 | FPR1_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (7VFX) | 7VFX | ||
| D0403 | DNA [cytosine-5]-methyltransferase 1 | P26358 | DNMT1_HUMAN | DNA methyltransferase | Clinical trial | Downloaded from PDB (6X9J) | 6X9J | ||
| D0404 | Erbb2 tyrosine kinase receptor | P04626 | ERBB2_HUMAN | transmembrane signal receptor | Successful | Downloaded from PDB (7PCD) | 7PCD | ||
| D0405 | Oxalosuccinate decarboxylase | O75874 | IDHC_HUMAN | dehydrogenase | Successful | Downloaded from PDB (4UMX) | 4UMX | ||
| D0406 | Neuropeptide Y receptor type 1 | P25929 | NPY1R_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (5ZBQ) | 5ZBQ | ||
| D0407 | C-C chemokine receptor type 2 | P41597 | CCR2_HUMAN | cell adhesion molecule | Clinical trial | Downloaded from PDB (6GPX) | 6GPX | ||
| D0408 | Programmed cell death 1 ligand 1 | Q9NZQ7 | PD1L1_HUMAN | immunoglobulin receptor superfamily | Successful | Downloaded from PDB (7NLD) | 7NLD | ||
| D0409 | Adenosine kinase | P55263 | ADK_HUMAN | Undefined | Clinical trial | Downloaded from PDB (2I6B) | 2I6B | ||
| D0410 | T-cell-specific kinase | Q08881 | ITK_HUMAN | non-receptor tyrosine protein kinase | Clinical trial | Downloaded from PDB (4M15) | 4M15 | ||
| D0411 | Angiopoietin 1 receptor | Q02763 | TIE2_HUMAN | transmembrane signal receptor | Clinical trial | Downloaded from PDB (6MWE) | 6MWE | ||
| D0412 | Lysophosphatidic acid receptor 1 | Q92633 | LPAR1_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (4Z35) | 4Z35 | ||
| D0413 | MALT lymphoma-associated translocation | Q9UDY8 | MALT1_HUMAN | cysteine protease | Clinical trial | Downloaded from PDB (7PAW) | 7PAW | ||
| D0414 | Presenilin 1 | P49768 | PSN1_HUMAN | aspartic protease | Clinical trial | Downloaded from PDB (7D8X) | 7D8X | ||
| D0415 | Ribosomal protein S6 kinase beta-1 | P23443 | KS6B1_HUMAN | protein modifying enzyme | Clinical trial | Downloaded from PDB (3WF7) | 3WF7 | ||
| D0416 | TYRO3 tyrosine kinase receptor | Q06418 | TYRO3_HUMAN | transmembrane signal receptor | Clinical trial | Modelled with AlphaFold (AF-Q06418-F1-model_v4) | AB INITIO | ||
| D0417 | Melanocortin receptor 5 | P33032 | MC5R_HUMAN | G-protein coupled receptor | Clinical trial | Modelled with SWISS-MODEL (7PIU.1.A) | HOMOLOGY | ||
| D0418 | Heat shock protein 90 beta | P08238 | HS90B_HUMAN | Hsp90 family chaperone | Clinical trial | Downloaded from PDB (5UCJ) | 5UCJ | ||
| D0419 | Fatty acid synthase | P49327 | FAS_HUMAN | Undefined | Successful | Downloaded from PDB (3HHD) | 3HHD | ||
| D0420 | Leucine-rich repeat kinase 2 | Q5S007 | LRRK2_HUMAN | scaffold/adaptor protein | Clinical trial | Downloaded from PDB (6OJF) | 6OJF | ||
| D0421 | MAPK signal-integrating kinase 1 | Q9BUB5 | MKNK1_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (2HW6) | 2HW6 | ||
| D0422 | ATM serine/threonine kinase | Q13315 | ATM_HUMAN | non-receptor serine/threonine protein kinase | Clinical trial | Downloaded from PDB (7NI4) | 7NI4 | ||
| D0423 | Fatty-acid amide hydrolase 1 | O00519 | FAAH1_HUMAN | hydrolase | Patented-recorded | Modelled with SWISSMODEL (3ppm.1.A) | HOMOLOGY | ||
| D0424 | Protein arginine methyltransferase 5 | O14744 | ANM5_HUMAN | protein modifying enzyme | Clinical trial | Downloaded from PDB (4X61) | 4X61 | ||
| D0425 | GABA | O14764 | GBRD_HUMAN | ligand-gated ion channel | Successful | Downloaded from PDB (7QNC) | 7QNC | ||
| D0426 | Lysine-specific demethylase 4A | O75164 | KDM4A_HUMAN | histone modifying enzyme | Patented-recorded | Downloaded from PDB (5VGI) | 5VGI | ||
| D0427 | Voltage-gated calcium channel alpha Cav3.2 | O95180 | CAC1H_HUMAN | voltage-gated ion channel | Successful | Modelled with AlphaFold (AF-O95180-F1-model_v6) | AB INITIO | ||
| D0428 | Influenza Polymerase acidic endonuclease | P03433 | PA_I34A1 | Undefined | Successful | Downloaded from PDB (5FDG) | 5FDG | ||
| D0429 | Lysosomal acid glucosylceramidase | P04062 | GBA1_HUMAN | Undefined | Clinical trial | Downloaded from PDB (9FB2) | 9FB2 | ||
| D0430 | Protein kinase C gamma | P05129 | KPCG_HUMAN | non-receptor serine/threonine protein kinase | Successful | Modelled with SWISSMODEL (8SE3.1.A) | HOMOLOGY | ||
| D0431 | Cholinesterase | P06276 | CHLE_HUMAN | esterase | Successful | Downloaded from PDB (6ZWI) | 6ZWI | ||
| D0432 | Matrix metalloproteinase-3 | P08254 | MMP3_HUMAN | metalloprotease | Patented-recorded | Downloaded from PDB (1HY7) | 1HY7 | ||
| D0433 | Bacterial DNA gyrase B | P0AES6 | GYRB_ECOLI | DNA topoisomerase | Clinical trial | Downloaded from PDB (7P2M) | 7P2M | ||
| D0434 | G2/mitotic-specific cyclin B1 | P14635 | CCNB1_HUMAN | kinase activator | Patented-recorded | Downloaded from PDB (6GU2) | 6GU2 | ||
| D0435 | Fatty acid-binding protein 4 | P15090 | FABP4_HUMAN | transfer/carrier protein | Patented-recorded | Downloaded from PDB (7FXV) | 7FXV | ||
| D0436 | Arachidonate 15-lipoxygenase | P16050 | LOX15_HUMAN | oxygenase | Patented-recorded | Modelled with SWISSMODEL (1lox.1.A) | HOMOLOGY | ||
| D0437 | Neuronal acetylcholine receptor beta-2 | P17787 | ACHB2_HUMAN | ligand-gated ion channel | Clinical trial | Downloaded from PDB (8ST4) | 8ST4 | ||
| D0438 | Galectin-3 | P17931 | LEG3_HUMAN | extracellular matrix protein | Clinical trial | Downloaded from PDB (7RH3) | 7RH3 | ||
| D0439 | Casein kinase II alpha prime | P19784 | CSK22_HUMAN | Undefined | Patented-recorded | Downloaded from PDB (6TEW) | 6TEW | ||
| D0440 | Adrenergic receptor alpha-1D | P25100 | ADA1D_HUMAN | G-protein coupled receptor | Successful | Modelled with AlphaFold (AF-P25100-F1-model_v6) | AB INITIO | ||
| D0441 | Proteasome beta-5 | P28074 | PSB5_HUMAN | protease | Patented-recorded | Downloaded from PDB (5L62) | 5L62 | ||
| D0442 | GABA | P31644 | GBRA5_HUMAN | ligand-gated ion channel | Successful | Downloaded from PDB (8BHG) | 8BHG | ||
| D0443 | Carbonic anhydrase VII | P43166 | CAH7_HUMAN | dehydratase | Patented-recorded | Downloaded from PDB (8Q3U) | 8Q3U | ||
| D0444 | Neuronal acetylcholine receptor alpha-4 | P43681 | ACHA4_HUMAN | ligand-gated ion channel | Successful | Downloaded from PDB (8ST4) | 8ST4 | ||
| D0445 | G-protein coupled receptor 6 | P46095 | GPR6_HUMAN | G-protein coupled receptor | Clinical trial | Downloaded from PDB (8T1V) | 8T1V | ||
| D0446 | Stress-activated protein kinase JNK3 | P53779 | MK10_HUMAN | non-receptor serine/threonine protein kinase | Patented-recorded | Downloaded from PDB (3OY1) | 3OY1 | ||
| D0447 | Phosphodiesterase 1B | Q01064 | PDE1B_HUMAN | phosphodiesterase | Patented-recorded | Downloaded from PDB (5UOY) | 5UOY | ||
| D0448 | Protein kinase C epsilon | Q02156 | KPCE_HUMAN | non-receptor serine/threonine protein kinase | Successful | Modelled with AlphaFold (AF-Q02156-F1-model_v6) | AB INITIO | ||
| D0449 | Phosphodiesterase 4C | Q08493 | PDE4C_HUMAN | phosphodiesterase | Patented-recorded | Downloaded from PDB (2QYM) | 2QYM | ||
| D0450 | Oxysterols receptor LXR-alpha | Q13133 | NR1H3_HUMAN | C4 zinc finger nuclear receptor | Patented-recorded | Downloaded from PDB (5HJS) | 5HJS | ||
| D0451 | Phosphodiesterase 3B | Q13370 | PDE3B_HUMAN | phosphodiesterase | Patented-recorded | Downloaded from PDB (1SO2) | 1SO2 | ||
| D0452 | Dual-specificity tyrosine-phosphorylation regulated kinase 1A | Q13627 | DYR1A_HUMAN | protein modifying enzyme | Patented-recorded | Downloaded from PDB (4YLK) | 4YLK | ||
| D0453 | Extracellular lysophospholipase D | Q13822 | ENPP2_HUMAN | hydrolase | Clinical trial | Downloaded from PDB (4ZG7) | 4ZG7 | ||
| D0454 | NAD-dependent deacetylase sirtuin-2 | Q8IXJ6 | SIR2_HUMAN | Undefined | Patented-recorded | Downloaded from PDB (9FDS) | 9FDS | ||
| D0455 | Histone deacetylase 7 | Q8WUI4 | HDAC7_HUMAN | Undefined | Patented-recorded | Downloaded from PDB (3C10) | 3C10 | ||
| D0456 | Growth hormone secretagogue receptor 1 | Q92847 | GHSR_HUMAN | G-protein coupled receptor | Successful | Downloaded from PDB (9UY3) | 9UY3 | ||
| D0457 | Histone deacetylase 10 | Q969S8 | HDA10_HUMAN | Undefined | Patented-recorded | Modelled with SWISSMODEL (7u59.1.A) | HOMOLOGY | ||
| D0458 | Histone deacetylase 11 | Q96DB2 | HDA11_HUMAN | Undefined | Patented-recorded | Modelled with AlphaFold (AF-Q96DB2-F1-model_v6) | AB INITIO | ||
| D0459 | Urate anion exchanger 1 | Q96S37 | S22AC_HUMAN | secondary carrier transporter | Successful | Downloaded from PDB (9DKC) | 9DKC | ||
| D0460 | Sphingosine-1-phosphate receptor 3 | Q99500 | S1PR3_HUMAN | G-protein coupled receptor | Patented-recorded | Downloaded from PDB (7EW2) | 7EW2 | ||
| D0461 | HIF-prolyl hydroxylase 2 | Q9GZT9 | EGLN1_HUMAN | Undefined | Patented-recorded | Downloaded from PDB (7Q5V) | 7Q5V | ||
| D0462 | Lysine-specific demethylase 4C | Q9H3R0 | KDM4C_HUMAN | histone modifying enzyme | Patented-recorded | Downloaded from PDB (5KR7) | 5KR7 | ||
| D0463 | Phosphatidylinositol-4-kinase beta | Q9UBF8 | PI4KB_HUMAN | kinase | Clinical trial | Downloaded from PDB (6GL3) | 6GL3 | ||
| D0464 | Histone deacetylase 9 | Q9UKV0 | HDAC9_HUMAN | Undefined | Patented-recorded | Modelled with AlphaFold (AF-Q9UKV0-6-F1-model_v6) | AB INITIO | ||
| D0465 | Histone deacetylase 5 | Q9UQL6 | HDAC5_HUMAN | Undefined | Patented-recorded | Modelled with AlphaFold (AF-Q9UQL6-3-F1-model_v6) | AB INITIO |
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